发明名称 PREPARATION OF 1-[4-(2-METHOXY-PHENYL)-PIPERAZIN-1-YL]-3-(2,6-DIOXOPIPERIDIN-1-YL) PROPANE HYDROCHLORIDE
摘要 <p>The present invention relates to processes for the synthesis of 1-[4-(2­methoxyphenyl)piperazin-1-yl]-3-(2,6-dioxopiperidin-1-yl) propane hydrochloride having protracted uro-selective (alpha1-adrenoceptor antagonistic activity. The compound holds promise for treating benign prostatic hyperplasia (BPH).</p>
申请公布号 WO2005021521(A1) 申请公布日期 2005.03.10
申请号 WO2003IB03585 申请日期 2003.08.28
申请人 RANBAXY LABORATORIES LIMITED;ANAND, NITYA;SINHA, NEELIMA;JAIN, SANJAY;MEHTA, ANITA 发明人 ANAND, NITYA;SINHA, NEELIMA;JAIN, SANJAY;MEHTA, ANITA
分类号 C07D213/69;(IPC1-7):C07D295/02 主分类号 C07D213/69
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