发明名称 Derivaten van piperazine.
摘要 This invention relates to a compound of formula (I) or pharmaceutically acceptable salts, solvates or derivatives thereof, wherein R<1> to R<5> are defined in the description, and to processes for the preparation thereof, intermediates used in their preparation, compositions containing them and the uses of such derivatives. The compounds of the present invention inhibit the interaction of gp 120 with CD4 and are therefore of use in the treatment of HIV, a retroviral infection genetically related to HIV, or AIDS.
申请公布号 NL1026827(A1) 申请公布日期 2005.03.09
申请号 NL20041026827 申请日期 2004.08.12
申请人 PFIZER INC. 发明人 DONALD STUART MIDDLETON;CHARLES ERIC MOWBRAY;PETER THOMAS STEPHENSON;DAVID HOWARD WILLIAMS
分类号 C07D213/64;C07D213/81;C07D215/20;C07D215/22;C07D215/227;C07D215/26;C07D215/38;C07D215/48;C07D217/02;C07D217/22;C07D217/24;C07D217/26;C07D231/12;C07D231/56;C07D233/54;C07D235/08;C07D239/74;C07D249/08;C07D263/56;C07D271/06;C07D295/192;C07D401/04;C07D401/12;(IPC1-7):C07D241/04;A61K31/496;A61P31/18;A61K31/470;C07D215/02;C07D261/20;C07D235/06;C07D271/10;C07D221/04 主分类号 C07D213/64
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