发明名称 |
OXAZOLIDINONE ANTIBIOTICS AND DERIVATIVES THEREOF |
摘要 |
<p>This invention relates to new oxazolidin,41-es having a C" cl ropyl moiety, which are effective against aerobic and anerobic pathogen I esistant staphylococci, streptococci and enterococci, Bacteroides s Cl' idia spp. species, as well as acid-fast organisms such as Mycobacterium tuberculosis and other mycobacterial species. 10 The compounds are represented by structural formula (I): A a Rx (R4a)s Rx x 1 0 Ri Ar or HAr N 0 A /_R3 15 its enantiomer, diastereomer, or pharmaceutically acceptable salt or ester thereof.</p> |
申请公布号 |
WO2005005399(A1) |
申请公布日期 |
2005.01.20 |
申请号 |
WO2004US20736 |
申请日期 |
2004.06.29 |
申请人 |
MERCK & CO., INC.;KYORIN PHARMACEUTICAL CO., LTD.;HAMMOND, MILTON, L.;FUKUDA, YASUMICHI |
发明人 |
HAMMOND, MILTON, L.;FUKUDA, YASUMICHI |
分类号 |
A61P31/04;C07D263/20;C07D413/06;C07D413/10;C07D413/14;C07F9/572;C07F9/6558;(IPC1-7):C07D263/20;C07F9/09;A61K31/422 |
主分类号 |
A61P31/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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