| 摘要 |
<p>A phenolic compound (I) is new. A phenolic compound of formula (I) is new. [Image] m : 0-2; R 1>, R 2>H, nitro, carboxyl, halogen, 1-6C alkyl, 1-6C alkoxy, 1-6C alkoxycarbonyl, sulfamoyl, phenylsulfamoyl, 1-6C alkylsulfamoyl, di-1-6C alkylsulfamoyl, carbamoyl, phenylcarbamoyl, 1-6C alkylcarbamoyl, di-1-6C alkylcarbamoyl, ureido, 1-6C alkylureido, di-1-6C alkylureido, tri-1-6C alkylureido or optionally substituted phenylureido; p, q : 0-4; t, u : 0 or 1 (both are not simultaneously 0); X : formula (II)-(VII); [Image] [Image] R 3>, R 4>, R 1> 0>, R 1> 1>H or 1-6C alkyl; R 5>H, 1-6C alkyl, optionally substituted phenyl, optionally substituted benzyl or formula (a); R 7>H, 1-6C alkyl, optionally substituted phenyl or optionally substituted benzyl; [Image] a : 1-6; Y 1>1-6C alkylene, formula (II') or formula (i)-(xvii); [Image] [Image] [Image] [Image] [Image] R 6>nitro, halogen, 1-6C alkyl, 1-6C alkoxy or 1-6C alkoxycarbonyl; b : 0-4; Y 2>single bond, CO or SO 2; Y 3>O or S; Y 4>CO or SO 2; Y 5>CO or NR 7>CO; R 8>, R 9>H, 1-6C alkyl or optionally substituted phenyl; c : 0-6; Y 6>single bond or (II'); Y 7>single bond or NH; Y 8>single bond or -SC(O)Y 7>Y 1>- (xvi). When X = (VI) or (VII), m = 0. When X = (II) or (VI), p, q = 0, t, u = 1, 2 OH's are para. When X = (III), (IV) or (VII), q = 0, u = 1, OH is para. When X = (VII), Y 8> = (xvi).</p> |
