发明名称 Carboxy pyrrole, process of preparing and use as precursor
摘要 4-Oxo-4,5-dihydro-3H-pyrrolo[3,2-d] pyrimidine-7-carboxylic acid methyl ester and process for preparing are provided. The 4-oxo-4,5-dihydro-3H-pyrrole[3,2-d] pyrimidine-7-carboxylic acid methyl ester is useful as a precursor for providing 9-deaza-hypoxanthine, a key intermediate for producing certain PNP inhibitors.
申请公布号 US2004214840(A1) 申请公布日期 2004.10.28
申请号 US20030420757 申请日期 2003.04.23
申请人 BIOCRYST PHARMACEUTICALS, INC. 发明人 WINSLOW CHRISTOPHER D.;MORRIS PHILIP E.
分类号 C07D487/04;(IPC1-7):A61K31/519;C07D487/02 主分类号 C07D487/04
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