发明名称 |
NOVEL METHOD FOR SYNTHESISING (2S, 3AS, 7AS)-PERHYDROINDOLE-2-CARBOXYLIC ACID AND THE ESTERS THEREOF AND THE USE THEREOF FOR PERINDOPRIL SYNTHESIS |
摘要 |
The invention relates to a method for synthesising derivatives of the formula (I), wherein R is a hydrogen atom or an amine function-protecting group. The use of said derivatives for synthesising perindopril and the pharmaceutically acceptable salts thereof is also disclosed. |
申请公布号 |
WO2004078707(A3) |
申请公布日期 |
2004.10.14 |
申请号 |
WO2004FR00444 |
申请日期 |
2004.02.27 |
申请人 |
LES LABORATOIRES SERVIER;DUBUFFET, THIERRY;LANGLOIS, PASCAL |
发明人 |
DUBUFFET, THIERRY;LANGLOIS, PASCAL |
分类号 |
C07D209/42 |
主分类号 |
C07D209/42 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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