发明名称 Peptide boronic acids useful in making salts thereof
摘要 <p>Tripeptide boronic acids of (R,S,R) configuration, for example Cbz-(R)-Phe-(S)-Pro-(R)-Mpg-B(OH)2, and their use to make base addition salts of such acids. The salts are formulated into antithrombotic pharmaceutical formulations.</p>
申请公布号 EP1466916(A1) 申请公布日期 2004.10.13
申请号 EP20040076510 申请日期 2003.09.09
申请人 TRIGEN LIMITED 发明人 MADGE, DAVID JONATHAN;DOLMAN, MARK;COMBE-MARZELLE, SOPHIE, MARIE;DEADMAN, JOHN, JOSEPH;KENNEDY, ANTHONY, JAMES;KAKKAR, SANJAY KUMAR;WALTER, ARMIN;OLBRICH, ALFRED;KRIMMER, DIETER;WEILAND-WEIBEL, ANDREA, MARIA, THERESIA
分类号 A61K31/69;A61K38/00;A61K45/06;C07F5/02;C07K5/06;C07K5/065;(IPC1-7):C07F5/02 主分类号 A61K31/69
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