发明名称 TRICYCLIC STEROID HORMONE NUCLEAR RECEPTOR MODULATORS
摘要 The present invention relates to methods of treating pathological disorders susceptible to steroid hormone nuclear receptor modulation comprising administering to a patient in need thereof an effective amount of a compound of the formula (I): or a pharmaceutically acceptable salt thereof. In addition, the present invention provides novel pharmaceutical compounds of Formula (I), including the pharmaceutically acceptable salts thereof, as well as pharmaceutical compositions which comprise as an active ingredient a compound of Formula (I).
申请公布号 WO2004052847(A3) 申请公布日期 2004.09.10
申请号 WO2003US16213 申请日期 2003.06.13
申请人 ELI LILLY AND COMPANY;COGHLAN, MICHAEL, JOSEPH;GREEN, JONATHAN, EDWARD;GRESE, TIMOTHY, ALAN;JADHAV, PRABHAKAR, KONDAJI;MATTHEWS, DONALD, PAUL;STEINBERG, MITCHELL, IRVIN;FALES, KEVIN, ROBERT;BELL, MICHAEL, GREGORY 发明人 COGHLAN, MICHAEL, JOSEPH;GREEN, JONATHAN, EDWARD;GRESE, TIMOTHY, ALAN;JADHAV, PRABHAKAR, KONDAJI;MATTHEWS, DONALD, PAUL;STEINBERG, MITCHELL, IRVIN;FALES, KEVIN, ROBERT;BELL, MICHAEL, GREGORY
分类号 C07D295/08;A61K31/015;A61K31/03;A61K31/04;A61K31/045;A61K31/055;A61K31/09;A61K31/10;A61K31/335;A61K31/381;A61K31/404;A61K31/415;A61K31/4164;A61K31/4184;A61K31/423;A61K31/428;A61K31/435;A61K31/4402;A61K31/4406;A61K31/4436;A61K31/4453;A61K31/4965;A61K31/5377;A61K31/55;A61P1/04;A61P1/16;A61P3/04;A61P3/08;A61P3/10;A61P3/12;A61P3/14;A61P5/26;A61P5/38;A61P5/46;A61P7/04;A61P7/10;A61P9/00;A61P9/02;A61P9/10;A61P9/12;A61P11/00;A61P11/06;A61P13/12;A61P17/00;A61P17/06;A61P17/10;A61P19/02;A61P19/10;A61P25/02;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P29/00;A61P35/00;A61P35/02;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07C22/04;C07C22/08;C07C25/22;C07C25/24;C07C33/38;C07C39/17;C07C39/23;C07C39/42;C07C43/215;C07C43/225;C07C43/23;C07C47/548;C07C47/57;C07C49/835;C07C205/06;C07C205/35;C07C211/32;C07C211/45;C07C215/76;C07C217/84;C07C233/07;C07C233/65;C07C233/84;C07C235/16;C07C251/40;C07C251/48;C07C255/50;C07C261/04;C07C271/14;C07C275/28;C07C307/10;C07C311/03;C07C311/08;C07C311/09;C07C311/16;C07C311/20;C07C311/21;C07C311/29;C07C317/14;C07C317/32;C07C321/28;C07C323/49;C07D209/08;C07D209/34;C07D211/18;C07D213/127;C07D213/16;C07D213/65;C07D213/73;C07D213/76;C07D213/81;C07D221/16;C07D223/20;C07D231/12;C07D231/18;C07D233/26;C07D233/64;C07D233/84;C07D235/26;C07D241/12;C07D241/20;C07D241/26;C07D261/08;C07D263/52;C07D263/56;C07D263/58;C07D277/60;C07D295/092;C07D295/22;C07D295/26;C07D313/14;C07D333/80;C07D337/12;C07D337/14;C07D401/06;C07D403/06;C07D405/04;C07D405/06;C07D409/04;C07D471/04;C07D487/04;C07D491/044 主分类号 C07D295/08
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