发明名称 PROCESS FOR THE SYNTHESIS OF INTERMEDIATES USEFUL FOR THE SYNTHESIS OF TUBULIN INHIBITORS
摘要 The invention is a process for the preparation of compounds of the Formula (I): where R1, R2, R3, R4 and R5 are defined in the specification, which are intermediates useful for the preparation of tubulin inhibitors useful in the treatment of cancer.
申请公布号 WO2004026814(A3) 申请公布日期 2004.08.12
申请号 WO2003US28661 申请日期 2003.09.12
申请人 WYETH HOLDINGS CORPORATION;WU, YANZHONG;MEGATI, SREENIVASULU;GLETSOS, CONSTANTINE;KENDALL, JOHN, THOMAS;WILK, BOGDAN, KAZIMIERZ;PADMANATHAN, THURAIRAJAH;RAVEENDRANATH, PANOLIL 发明人 WU, YANZHONG;MEGATI, SREENIVASULU;GLETSOS, CONSTANTINE;KENDALL, JOHN, THOMAS;WILK, BOGDAN, KAZIMIERZ;PADMANATHAN, THURAIRAJAH;RAVEENDRANATH, PANOLIL
分类号 A61K38/00;C07C45/44;C07C45/58;C07C231/18;C07C237/22;C07C269/08;C07C271/22;C07C313/06;C07K5/02 主分类号 A61K38/00
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