供作药剂之新颖胺基唑衍生物及包含其之医药组合物(二) NOVEL AMINOINDAZOLE DERIVATIVES AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS INCLUDING THEM

摘要

本发明有关一种具有通式(I)之新颖衍生物092124408p01.bmp其中R3系为(1–6C)烷基、芳基、芳基(1–6C)烷基、杂芳基、杂芳基(1–6C)烷基、稠合于(1–10C)环烷基之芳基或杂芳基、杂环、杂环烷基、环烷基、金刚烷基、多环烷基、烯基、炔基、CONR1R2、COOR1、SO2R1、C(＝NH)R1或C(＝NH)NR1基团；R5及R6个别选自下列基团：卤素、CN、NO2、NH2、OH、COOH、C(O)OR8、–O–C(O)R8、NR8R9、NHC(O)R8、C(O)NR8R9、NHC(S)R8、C(S)NR8R9、SR8、S(O)R8、SO2R8、NHSO2R8、SO2NR8R9、–O–SO2R8、–SO2–O–R8、三氟甲基、三氟甲氧基、(1–6C)烷基、(1–6C)烷氧基、芳基、芳基(1–6C)烷基、杂芳基、杂芳基(1–6C)烷基、杂环、环烷基、烯基、炔基、金刚烷基或多环烷基。092124408p01.bmp