发明名称 |
1,2,4-TRIAZIN-3-YL-HYDRAZINE OR 5H-1,2,4-TRIAZINO'5,6-B!INDOL-3-YL-HYDRAZINE COMPOUNDS AS INHIBITORS OF BACE USEFUL IN THE TREATMENT OF ALZHEIMER |
摘要 |
<p>A compound of formula (I) wherein R<1> is aryl and R<2> is hydrogen; or R<1> and R<2> taken together form a group of formula (i) wherein R<6> is alkyl or -alkyl-aryl; and R<7> is hydrogen, halogen, alkyl, alkoxy or aryl; R<3> is aryl, heteroaryl or -aryl-aryl; R<4> is hydrogen, hydroxy or alkyl; and R<5> is hydrogen or alkyl; or a pharmaceutically acceptable salt thereof, is new, for use in therapy, e.g. of Alzheimer's disease.</p> |
申请公布号 |
WO2004063196(A1) |
申请公布日期 |
2004.07.29 |
申请号 |
WO2004GB00062 |
申请日期 |
2004.01.12 |
申请人 |
DE NOVO PHARMACEUTICALS LIMITED;WILLEMS, HENRIETTE;HARRIS, WILLIAM;JOHN, DEREK, EDWARD |
发明人 |
WILLEMS, HENRIETTE;HARRIS, WILLIAM;JOHN, DEREK, EDWARD |
分类号 |
A61P25/28;C07D403/12;C07D487/04;(IPC1-7):C07D487/04;A61K31/53 |
主分类号 |
A61P25/28 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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