发明名称 (2-CARBOXAMIDO) (3-AMINO) THIOPHENE COMPOUNDS
摘要 Compounds represented by Formula (I): or a pharmaceutically acceptable salt or N-oxide thereof, wherein R1 is R2;< >and R3 is C0-4 alkyl, are useful in the treatment of cancer.
申请公布号 WO2004063330(A2) 申请公布日期 2004.07.29
申请号 WO2004US01188 申请日期 2004.01.06
申请人 OSI PHARMACEUTICALS, INC.;WYNNE, GRAHAM, MICHAEL;DOYLE, KEVIN;AHMED, SALEH;LI, AN-HU;KEILY, JOHN FRASER;RASAMISON, CHRYSTELLE;PEGG, NEIL ANTHONY;SABA, IMAAD;THOMAS, CLAIRE;SMYTH, DON;SADIQ, SHAZIA;NEWTON, GARY;DAWSON, GRAHAM;CREW, ANDREW PHILIP;CASTELANO, ARLINDO LUCAS 发明人 WYNNE, GRAHAM, MICHAEL;DOYLE, KEVIN;AHMED, SALEH;LI, AN-HU;KEILY, JOHN FRASER;RASAMISON, CHRYSTELLE;PEGG, NEIL ANTHONY;SABA, IMAAD;THOMAS, CLAIRE;SMYTH, DON;SADIQ, SHAZIA;NEWTON, GARY;DAWSON, GRAHAM;CREW, ANDREW PHILIP;CASTELANO, ARLINDO LUCAS
分类号 A61K31/381;A61K31/437;A61K31/4436;A61K31/4709;A61K31/4745;A61K45/06;C07D409/12;C07D409/14;C07D471/04 主分类号 A61K31/381
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