发明名称 Process and intermediates for making non-nucleoside HIV-1 reverse transcriptase inhibitors
摘要 A process and novel intermediates for making compounds of the formula I:wherein:R<2 >is selected from the group consisting of H, F, Cl, C1-4 alkyl, C3-4 cycloalkyl and CF3;R<4 >is H or Me;R<5 >is H, Me or Et, with the proviso that R<4 >and R<5 >are not both Me, and if R<4 >is Me then R<5 >cannot be Et;R<11 >is Me, Et, cyclopropyl, propyl, isopropyl, or cyclobutyl; andQ is selected from the group consisting of:
申请公布号 US6759533(B2) 申请公布日期 2004.07.06
申请号 US20030465754 申请日期 2003.06.19
申请人 BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 发明人 BUSACCA CARL A.;ERIKSSON MAGNUS C.;KIM JI-YOUNG
分类号 C07D471/04;C07B61/00;C07D471/14;C07F9/6524;(IPC1-7):C07D471/14 主分类号 C07D471/04
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