发明名称 Indolylpiperidine derivatives as antihistaminic aand antiallergic agents
摘要 The invention relates to indolyl piperidinyl derivatives of formula (I) wherein: A<1 >represents an alkylene, alkyleneoxy, alkylenethio, alkanoylene or hydroxyalkylene group; A<2 >represents an alkylene, alkyleneoxy, alkylenethio, alkanoylene or an alkyleneoxyalkylene group; W<1 >represents a phenylene, furanylene or pyridinylene group which is unsubstituted or substituted by one or more halogen atoms, alkoxy groups and/or alkyl groups; W<2 >represents a 3-10 membered monocyclic or bicyclic group containing from 1 to 3 heteroatoms said group being unsubstituted or substituted by one or more halogen atoms, alkyl groups, alkoxy groups and/or oxo groups; R<1 >represents a hydrogen or halogen atom or an alkyl, alkoxy or methylamino group; and R<2 >represents a carboxyl group; and pharmaceutically acceptable salts thereof; to processes for their preparation; to pharmaceutical compositions containing them; and to their medical use as antihistaminic and antiallergic agents.
申请公布号 US2004116471(A1) 申请公布日期 2004.06.17
申请号 US20030415693 申请日期 2003.12.16
申请人 POU SILVIA FONQUERNA;PAGES SANTACANA LLUIS;PUIG DURAN CARLES;SOCA PUEYO LIDIA 发明人 POU SILVIA FONQUERNA;PAGES SANTACANA LLUIS;PUIG DURAN CARLES;SOCA PUEYO LIDIA
分类号 C07D401/04;A61K31/454;A61K31/4545;A61K31/5377;A61P11/06;A61P17/00;A61P27/02;A61P27/16;A61P37/08;A61P43/00;C07D401/14;C07D405/14;C07D409/14;C07D413/14;(IPC1-7):A61K31/454;C0741/14 主分类号 C07D401/04
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