发明名称 CRYSTALLINE 17BETA-HYDROXY-7ALPHA- (5'-METHYL-2'-FURYL)-PREGNA-4,9(11)-DIEN-3-ONE-21-CARBOXYLIC ACID, GAMMA-LACTONE
摘要 The present invention involves a novel crystal form of 17beta-hydroxy-7alpha-(5'-methyl-2'-furyl)-pregna-4,9(11)-dien-3-one-21-carboxylic acid, gamma-lactone (II) which is an intermediate useful in preparation of an important pharmaceutical, eplerenone. (FORMULA)
申请公布号 WO2004037844(A8) 申请公布日期 2004.06.10
申请号 WO2003US29923 申请日期 2003.09.19
申请人 PHARMACIA & UPJOHN COMPANY;PEARLMAN, BRUCE, ALLEN;ANTOSZ, FREDERICK, J. 发明人 PEARLMAN, BRUCE, ALLEN;ANTOSZ, FREDERICK, J.
分类号 A61K31/58;C07J1/00;C07J21/00;(IPC1-7):C07J21/00 主分类号 A61K31/58
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