发明名称 |
METHODS OF TREATING CANCER AND RELATED METHODS |
摘要 |
Methods of treating cancer using 4-amino-5-fluoro-3-[6-(4-methylpiperazin-1- yl)-1H-benzimidazol-2-yl]quinolin-2(1H)-one are provided. In particular, the methods are effective for the treatment of solid tumors or leukemias, including prostate, colorectal, breast, multiple myeloma, pancreatic, small cell carcinoma, acute myelogenous leukemia, chronic myelogenous leukemia, or myelo-proliferative disease. Further provided are methods of measuring the amount of 4-amino-5-fluoro-3-[6-(4-methylpiperazin-1-yl)-1H-benzimidazol-2- yl]quinolin-2(1H)-one and determining a metabolic profile therefore.
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申请公布号 |
CA2501932(A1) |
申请公布日期 |
2004.05.27 |
申请号 |
CA20032501932 |
申请日期 |
2003.11.12 |
申请人 |
CHIRON CORPORATION |
发明人 |
ZHU, SHUGUANG;HARWOOD, ERIC;HAROLDSEN, PETER;SHANG, XIAO;HEISE, CARLA C.;SAMARA, EMIL;HANNAH, ALISON;VORA, JAYESH;MACHAJEWSKI, TIMOTHY D. |
分类号 |
A61K9/00;A61K31/4375;A61K31/4709;A61K31/496;A61K31/52;A61K47/26;A61P35/00;C07D401/04;C07D401/14;C07D405/14;C07D409/14;C07D413/14;C07D453/02;C07D453/06;C07D471/04;(IPC1-7):A61K31/496 |
主分类号 |
A61K9/00 |
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