发明名称 |
DERIVATIVES OF [6,7-DIHYDRO-5H-IMIDAZO[1,2-alpha]IMIDAZOLE-3-SULFONYL]-PYRROLIDINE-2-CARBOXYLIC ACID AMIDE AS ANTI-INFLAMMATORY AGENTS |
摘要 |
<p>Derivatives of 6,7-dihydro-5H-imidazo[1,2-alpha]imidazole-3-sulfonyl]-pyrrolidine-2-carboxylic acid amide which exhibit good inhibitory effect upon the interaction of CAMs and Leukointegrins and are thus useful in the treatment of inflammatory disease.</p> |
申请公布号 |
WO2004041273(A1) |
申请公布日期 |
2004.05.21 |
申请号 |
WO2003US33966 |
申请日期 |
2003.10.27 |
申请人 |
BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. |
发明人 |
KELLY, TERENCE, ALFRED;KIM, JIN, MI;LEMIEUX, RENE, MARC;TSCHANTZ, MATT, AARON |
分类号 |
A61K31/4166;A61K31/4188;A61K31/5375;A61P29/00;C07D235/02;C07D403/12;C07D413/02;C07D487/04;(IPC1-7):A61K31/418 |
主分类号 |
A61K31/4166 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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