发明名称 CONTINUOUS PROCESS FOR THE PREPARATION OF FRUCTOPYRANOSE SULFAMATE DERIVATIVES
摘要 <p>The present invention is directed to a continuous process for the preparation of fructopyranose sulfamate derivatives of the general formula (I) wherein R&lt;1&gt;, R&lt;3&gt;, R&lt;4&gt;, R&lt;5&gt;, R&lt;6&gt; and X are as herein defined. The present invention is further directed to a continuous process for the preparation of Topiramate.</p>
申请公布号 WO2004041836(A1) 申请公布日期 2004.05.21
申请号 WO2003US34107 申请日期 2003.10.27
申请人 ORTHO-MCNEIL PHARMACEUTICAL, INC. 发明人 ADKINS, THOMAS, W.;CICCO, CHARLES, F.;FEIBUSH, PENINA;KOCH, DONALD, A.;MARYANOFF, CYNTHIA;STALZER, WALTER, E.
分类号 C07D317/44;C07D493/02;C07D493/04;C07H;C07H9/04;C07H11/00;(IPC1-7):C07H11/00 主分类号 C07D317/44
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