发明名称 BENZOTHIENYL ANALOGUE OF SOMATOSTATIN, SELECTIVE FOR CERTAIN SOMATOSTATIN RECEPTORS
摘要 The invention relates to a peptide compound having an improved binding affinity to somatostatin receptors, comprising a peptide and a chelating group covalently linked to a free amino group of said peptide, wherein said peptide is or comprises a somatostatin analogue carrying a 3-benzothienylalanine residue in its 3-position. The invention further relates to said peptide compound labelled with a detectable element or with a therapeutic radionuclide, as well as to a diagnostic method and to a method for the therapeutic treatment of tumors, by using the labelled compounds.
申请公布号 WO03092744(A3) 申请公布日期 2004.04.01
申请号 WO2003EP04847 申请日期 2003.05.02
申请人 BIOSYNTHEMA INC.;MAECKE, HELMUT, ROBERT;REUBI, JEAN, CLAUDE;DE JONG, MARION;KRENNING, ERIC, PAUL;GINJ, MIHAELA 发明人 MAECKE, HELMUT, ROBERT;REUBI, JEAN, CLAUDE;DE JONG, MARION;KRENNING, ERIC, PAUL;GINJ, MIHAELA
分类号 A61K51/08 主分类号 A61K51/08
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