发明名称 |
alpha-Substituted beta-aminoethyl phosphonate derivatives |
摘要 |
The present invention relates to novel alpha-substituted-beta-aminoethylphosphonate and alpha-substituted-beta-aminovinylphosphonate derivatives and their uses for lowering plasma levels of apo (a), Lp(a), apo B, apo B associated lipoproteins (low density lipoproteins and very low density lipoproteins) and for lowering plasma levels of total cholesterol.
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申请公布号 |
US6706698(B2) |
申请公布日期 |
2004.03.16 |
申请号 |
US20010963900 |
申请日期 |
2001.09.26 |
申请人 |
ILEX PRODUCTS, INC. |
发明人 |
PHAN HIEU TRUNG;NGUYEN LAN MONG;DIEP VINH VAN;AZOULAY RAYMOND;ESCHENHOF HARALD;NIESOR ERIC JOSEPH;BENTZEN CRAIG LEIGH;IFE ROBERT JOHN |
分类号 |
A61K31/662;A61K31/675;A61P3/06;A61P7/02;A61P9/10;C07F9/58;C07F9/59;C07F9/6509;C07F9/6512;C07F9/6539;C07F9/6541;(IPC1-7):A01N57/00;C07F9/02;C07F9/06 |
主分类号 |
A61K31/662 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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