发明名称 METHOD FOR THE SELECTIVE PREPARATION OF 3-OXO-4-AZA-5A-ANDROSTANE COMPOUND
摘要 This invention relates to a method for selectively preparing the 3-oxo-4-aza-5¥á-androstane compound which is used as an intermediate of finasteride by heating 3-oxo-4-aza-5-androstene in a mixture of formic acid and an alkanediol in the presence of zinc.
申请公布号 WO2004016595(A1) 申请公布日期 2004.02.26
申请号 WO2003KR01629 申请日期 2003.08.13
申请人 HANMI PHARM. CO., LTD.;MOON, YOUNG-HO;LEE, KYUNG-IK;PARK, GHA-SEUNG;PARK, CHUL-HYUN;LEE, JAE-CHEOL;LEE, GWAN-SUN;CHANG, YOUNG-KIL 发明人 MOON, YOUNG-HO;LEE, KYUNG-IK;PARK, GHA-SEUNG;PARK, CHUL-HYUN;LEE, JAE-CHEOL;LEE, GWAN-SUN;CHANG, YOUNG-KIL
分类号 C07D221/18;C07J73/00 主分类号 C07D221/18
代理机构 代理人
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