发明名称 |
Indolylpiperidine derivatives as antihistaminic and antiallergic agents |
摘要 |
Indolylpiperidine compounds of formula (I)wherein:A<1 >represents an alkylene, alkyleneoxy, alkylenethio, alkanoyl or hydroxyalkylene group;A<2 >represents a single bond, an alkylene or alkenylene group;W represents a single bond or a phenylene or furanylene group which is unsubstituted or substituted by one or more halogen atoms, alkoxy groups and/or alkyl groups;R<2 >represents a hydrogen or halogen atom or an alkyl or alkoxy group; andR<3 >represents a carboxyl group or a tetrazolyl group.The present invention provides novel indolylpiperidine compounds having imporved antihistamine and antiallergic activity.
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申请公布号 |
US6683096(B2) |
申请公布日期 |
2004.01.27 |
申请号 |
US20010006416 |
申请日期 |
2001.12.04 |
申请人 |
ALMIRALL PRODESFARMA, S.A. |
发明人 |
PAGES SANTACANA LLUIS;FONQUERNA POU SILVIA;PUIG DURAN CARLES;FERNANDEZ FORNER MARIA DOLORS |
分类号 |
A61K31/445;A61K31/4525;A61K31/454;A61P11/02;A61P11/04;A61P11/06;A61P27/02;A61P37/08;C07D401/04;C07D401/14;C07D405/14;(IPC1-7):A61K31/445 |
主分类号 |
A61K31/445 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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