发明名称 Amidino and guanidino azetidinone derivatives useful as tryptase inhibitors
摘要 A beta lactam compounds of formulas (I), (IV) and (V) for use as inhibitors of various enzyme systems including tryptase, thrombin, trypsin, Factor Xa, Factor VIIa and urokinase type-plasminogen activator.
申请公布号 NZ507627(A) 申请公布日期 2003.12.19
申请号 NZ19990507627 申请日期 1999.06.18
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 BISACCHI, GREGORY;SLUSARCHYK, WILLIAM A;TREUNER, UWE;UTTON, JAMES C;ZAHLER, ROBERT;SEILER, STEVEN;KRONENTHAL,DAVID R;RANDAZZO, MICHAEL E;XU, ZHONGMIN;SHI, ZHONGPING;CHWINDEN, MARK D
分类号 A61K31/195;A61K31/397;A61K31/4025;A61K31/4427;A61K31/4433;A61K31/4523;A61K31/4725;A61K31/496;A61K31/506;A61K31/551;A61P11/00;A61P11/02;A61P11/06;A61P29/00;A61P43/00;C07D205/08;C07D205/09;C07D401/06;C07D401/12;C07D401/14;C07D403/06;C07D403/12;C07D409/06;(IPC1-7):C07D205/08 主分类号 A61K31/195
代理机构 代理人
主权项
地址