Amidino and guanidino azetidinone derivatives useful as tryptase inhibitors
摘要
A beta lactam compounds of formulas (I), (IV) and (V) for use as inhibitors of various enzyme systems including tryptase, thrombin, trypsin, Factor Xa, Factor VIIa and urokinase type-plasminogen activator.
申请公布号
NZ507627(A)
申请公布日期
2003.12.19
申请号
NZ19990507627
申请日期
1999.06.18
申请人
BRISTOL-MYERS SQUIBB COMPANY
发明人
BISACCHI, GREGORY;SLUSARCHYK, WILLIAM A;TREUNER, UWE;UTTON, JAMES C;ZAHLER, ROBERT;SEILER, STEVEN;KRONENTHAL,DAVID R;RANDAZZO, MICHAEL E;XU, ZHONGMIN;SHI, ZHONGPING;CHWINDEN, MARK D