发明名称 Crystalline fluoroquinolone arginine salt form
摘要 The invention relates to the new arginine salt forms of RS-(±)-9-fluoro-6,7-dihydro-8-(4-hydroxypiperidin-1-yl)-5-methyl-1-oxo-1H,5H-benzo[i,j]quinolizine-2-carboxylic acid, S-(-)-9-fluoro-6,7-dihydro-8-(4-hydroxypiperidin-1-yl)-5-methyl-1-oxo-1H,5H-benzo[i,j]quinolizine-2-carboxylic acid, R-(+)-9-fluoro-6,7-dihydro-8-(4-hydroxypiperidin-1-yl)-5-methyl-1-oxo-1H,5H-benzo[i,j]quinolizine-2-carboxylic acid, a process for their preparation and pharmaceutical formulations which comprise those arginine salt forms as the active ingredient for its use in treating microbial infections.
申请公布号 US6664267(B1) 申请公布日期 2003.12.16
申请号 US20020156685 申请日期 2002.05.28
申请人 WOCKHARDT LIMITED 发明人 DE SOUZA NOEL J.;DESHPANDE PRASAD K;SHUKLA MILIND C.;JAWEED MUKARRAM SIDDIQUI M;KULKARNI DILIP GANESH;RAHMAN ANSARI AZIZUR;YEOLE RAVINDRA D;PATEL MAHESH V;GUPTE SHRIKANT V
分类号 A61P31/04;C07D455/04;(IPC1-7):C07D455/04;A61K31/437 主分类号 A61P31/04
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