发明名称 |
3(5)-UREIDO-PYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS |
摘要 |
3-ureido-pyrazole derivatives represented by formula (I):where R, R1 and R2 are as described herein, or pharmnaceutically acceptable salts thereof; are useful, for example, for the treatment of cancer, cell proliferative disorders, Alzheimer's disease, viral infections, auto-immune diseases or neurodegenerative diseases. |
申请公布号 |
PL354058(A1) |
申请公布日期 |
2003.12.15 |
申请号 |
PL20000354058 |
申请日期 |
2000.08.11 |
申请人 |
PHARMACIA & UPJOHN SPA.;PHARMACIA & UPJOHN CO. |
发明人 |
PEVARELLO PAOLO;ORSINI PAOLO;TRAQUANDI GABRIELLA;VARASI MARIO;FRITZEN EDWARD L.;WARPEHOSKI MARTHA A.;PIERCE BETSY S. |
分类号 |
C07D231/38;A61K31/415;A61K31/4155;A61K31/4178;A61K31/428;A61K31/4439;A61K31/454;A61K31/4725;A61K31/496;A61K31/498;A61K31/5377;A61P9/10;A61P11/00;A61P13/12;A61P17/06;A61P19/02;A61P35/00;A61P35/02;C07D231/16;C07D231/40;C07D403/12 |
主分类号 |
C07D231/38 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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