发明名称 Piperidyindoles as serotonin receptor ligands
摘要 A pharmaceutical compound of the formula (I) in which R<1 >and R<2 >are each hydrogen or C1-6 alkyl, R<3 >is -SR<10>, -SOR<10>, -SO2R<10>, -COR<10>, -CH2OH or -CONHR<11>, where R<10 >is C1-6 alkyl and R<11 >is hydrogen or C1-6 alkyl, R<4>, R<5>, R<6 >and R<7 >are each hydrogen or C1-6 alkyl, provided that at least one of R<4>, R<5>, R<6 >and R<7 >is C1-6 alkyl, R<8 >and R<9 >are each hydrogen, halo, C1-6 alkyl or cyano, n is 0 or 1 and m is 2 or 3, x is a (a) or (b), and y is (c) or (d), wherein R<12 >and R<13 >are each hydrogen, C1- alkyl, cyclopropyl or cyclopropyl-C1-6 alkyl; and salts thereof.
申请公布号 US2003225068(A1) 申请公布日期 2003.12.04
申请号 US20020258356 申请日期 2002.10.21
申请人 FAIRHURST JOHN;GALLAGHER PETER 发明人 FAIRHURST JOHN;GALLAGHER PETER
分类号 A61P25/24;C07D401/14;C07D417/14;(IPC1-7):C07D417/14;A61K31/549 主分类号 A61P25/24
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