发明名称 AMINOQUINOLINE AND AMINOPYRIDINE DERIVATIVES AND THEIR USE AS ADENOSINE A3 LIGANDS
摘要 Compounds of general formula (I), wherein R<4> and R<5> stand for hydrogen atom or form together an 1,3-butadienyl group, optionally substituted by a methylenedioxy group or one or more straight or branched C1-4 alkyl group, straight or branched C1-4 alkoxy group, hydroxy group or halogen atom; are strong adenosine A3 receptor ligands preferably antagonists.
申请公布号 WO02096879(A9) 申请公布日期 2003.11.20
申请号 WO2002HU00048 申请日期 2002.05.29
申请人 SANOFI-SYNTHELABO;ARANYI, PETER;BALAZS, LASZLO;BALOGH, MARIA;BATA, IMRE;BATORI, SANDOR;T. NAGY, LAJOS;TIMARI, GEZA;BOER, KINGA;FINANCE, OLIVIER;KAPUI, ZOLTAN;MIKUS, ENDRE;SZAMOSVOELGYI, ZSUZSANNA;SZELECZKY, GABOR;URBAN-SZABO, KATALIN 发明人 ARANYI, PETER;BALAZS, LASZLO;BALOGH, MARIA;BATA, IMRE;BATORI, SANDOR;T. NAGY, LAJOS;TIMARI, GEZA;BOER, KINGA;FINANCE, OLIVIER;KAPUI, ZOLTAN;MIKUS, ENDRE;SZAMOSVOELGYI, ZSUZSANNA;SZELECZKY, GABOR;URBAN-SZABO, KATALIN
分类号 C07D215/54;A61K;A61K31/4706;A61K31/4709;A61P;A61P3/10;A61P9/00;A61P9/10;A61P9/12;A61P11/00;A61P11/06;A61P13/12;A61P17/06;A61P25/00;A61P25/16;A61P25/24;A61P27/06;A61P29/00;A61P35/00;A61P37/08;A61P43/00;C07D;C07D213/75;C07D213/85;C07D215/46;C07D215/48;C07D401/12;C07D405/12;C07D405/14;C07D409/12;C07D409/14 主分类号 C07D215/54
代理机构 代理人
主权项
地址