发明名称 |
MEDICINAL COMPOSITIONS IMPROVED IN SOLUBLITY IN WATER |
摘要 |
<p>Solid dispersions are provided comprising an HER2 inhibitor which is hardly or not soluble in water and a hydrophilic polymer. These solid dispersions have been improved in the solubility of the HER2 inhibitor, oral absorption and bioavailability in blood.</p> |
申请公布号 |
EP1350792(A1) |
申请公布日期 |
2003.10.08 |
申请号 |
EP20010270217 |
申请日期 |
2001.12.10 |
申请人 |
TAKEDA CHEMICAL INDUSTRIES, LTD. |
发明人 |
AKIYAMA, YOHKO;IINUMA, SATOSHI;BANDO, HIROTO |
分类号 |
A61K9/14;A61K9/16;A61K9/20;A61P35/00;C07D413/12;(IPC1-7):C07D413/12;A61K47/40;A61K47/38;A61K47/32;A61K47/28;A61K47/20;A61K9/10;A61K31/422;A61K47/26 |
主分类号 |
A61K9/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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