发明名称 Processes and intermediates for preparing glycogen phosphorylase inhibitors
摘要 The instant invention provides novel processes and intermediates useful in the preparation of certain N-(indole-2-carbonyl)-beta-alaninamide compounds, which compounds are glycogen phosphorylase inhibitors useful in the treatment of diseases such as hypercholesterolemia, hyperglycemia, hyperinsulinemia, hyperlipidemia, hypertension, atherosclerosis, diabetes, diabetic cardiomyopathy, infection, tissue ischemia, myocardial ischemia, and in inhibiting tumor growth.
申请公布号 US2003187051(A1) 申请公布日期 2003.10.02
申请号 US20030345661 申请日期 2003.01.16
申请人 PFIZER INC. 发明人 BARRILA MARK T.;BUSCH FRANK R.;COUTURIER MICHEL A.;ORRILL SUSAN L.;ROSE PETER R.;TICKNER DEREK L.;TOBIASSEN HARRY O;WITHBROE GREGORY J.
分类号 C07D491/056;C07D403/12;C07D491/04;(IPC1-7):A61K31/405;C0743/02 主分类号 C07D491/056
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