发明名称 Cyclic amino acid derivatives
摘要 Novel compounds of the formula I in which R1, R2, R2', R2'', R3, R4, R5, R5', R5'', R5''', R5'''', X, Y, U, V and W are as defined in Patent claim 1, are inhibitors of coagulation factors Xa and VIIa and can be employed fr the treatment of thromboses, myocardilal infarction, arteriosclerosis, inflammation, apoplexia, angina pectoris, restenosis after angioplasty, claudicatio intermittens, tumours, tumour diseases and/or tumour metastases.
申请公布号 US2003176465(A1) 申请公布日期 2003.09.18
申请号 US20030333278 申请日期 2003.01.17
申请人 MEDERSKI WERNER;JURASZYK HORST;DORSCH DIETER;TSAKLAKIDIS CHRISTOS;GLEITZ JOHANNES;BARNES CHRISTOPHER 发明人 MEDERSKI WERNER;JURASZYK HORST;DORSCH DIETER;TSAKLAKIDIS CHRISTOS;GLEITZ JOHANNES;BARNES CHRISTOPHER
分类号 C07D295/20;A61K31/397;A61K31/402;A61K31/4166;A61K31/421;A61K31/426;A61K31/4439;A61K31/451;A61K31/495;A61K45/00;A61P7/02;A61P7/04;A61P9/00;A61P9/10;A61P25/00;A61P29/00;A61P35/00;A61P43/00;C07D205/04;C07D207/16;C07D207/28;C07D211/34;C07D211/60;C07D233/34;C07D233/36;C07D263/06;C07D263/24;C07D277/06;C07D401/04;C07D413/12;(IPC1-7):A61K31/443;C07D413/02;C07D213/42;C07D213/57;C07D213/53;A61K31/44 主分类号 C07D295/20
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