发明名称 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR
摘要 Compounds of formula (I), are novel VR1 antagonists that are useful in treating pain, inflammatory thermal hyperalgesia, urinary incontinence and bladder overactivity.
申请公布号 WO03070247(A1) 申请公布日期 2003.08.28
申请号 WO2003US04187 申请日期 2003.02.11
申请人 ABBOTT LABORATORIES 发明人 LEE, CHIH-HUNG;BAYBURT, EROL, K.;DIDOMENICO, STANLEY, JR.;DRIZIN, IRENE;GOMTSYAN, ARTHUR, R.;KOENIG, JOHN, R.;PERNER, RICHARD, J.;SCHMIDT, ROBERT, G.;TURNER, SEAN, C.;WHITE, TAMMIE, K.;ZHENG, GUO, ZHU
分类号 A61K31/404;A61K31/416;A61K31/47;A61K31/472;A61K31/496;A61K31/5377;A61K31/541;C07D209/08;C07D217/02;C07D217/22;C07D217/24;C07D217/26;C07D231/56;C07D237/28;C07D401/12;C07D405/12;C07D521/00;(IPC1-7):A61K31/502 主分类号 A61K31/404
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