发明名称 N-BIPHENYLMETHYL AMINOCYCLOALKANECARBOXAMIDE DERIVATIVES WITH A SUBSTIITUENT ON THE METHYL USEFUL AS BRADYKININ ANTAGONISTS
摘要 N-Biphenyl(substituted methyl)aminocycloalkanecarboxamide derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
申请公布号 CA2474373(A1) 申请公布日期 2003.08.14
申请号 CA20032474373 申请日期 2003.02.04
申请人 MERCK & CO., INC. 发明人 KUDUK, SCOTT D.;FENG, DONG-MEI;WAI, JENNY MIU-CHUN;SU, DAI-SHI;ANTHONY, NEVILLE J.;BOCK, MARK G.;WOOD, MICHAEL R.
分类号 A61K31/166;A61K31/24;A61K31/41;A61K31/42;A61K31/4245;A61K31/505;A61P1/02;A61P1/04;A61P1/16;A61P1/18;A61P9/10;A61P11/00;A61P11/06;A61P11/08;A61P13/10;A61P13/12;A61P17/02;A61P17/06;A61P19/02;A61P19/08;A61P21/00;A61P25/04;A61P25/06;A61P25/28;A61P27/16;A61P29/00;A61P31/04;A61P35/00;A61P37/08;C07C237/24;C07D213/82;C07D239/28;C07D257/04;C07D261/18;C07D271/06;C07D403/12;C07D413/12;(IPC1-7):C07C237/24;C07D239/00;C07D261/00;C07D271/00 主分类号 A61K31/166
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