| 发明名称 |
AMIDES OF AMINOALKYL-SUBSTITUTED AZETIDINES, PYRROLIDINES, PIPERIDINES AND AZEPANES |
| 摘要 |
Novel amides of aminoalkyl-substituted azetidines, pyrrolidines, piperidines and azepanes, use of these compounds as pharmaceutical compositions, pharmaceutical compositions comprising the compounds, and a method of treatment employing these compounds and compositions. The compounds show a high and selective binding affinity to the histamine H3 receptor indicating histamine H3 receptor antagonistic, inverse agonistic or agonistic activity. As a result, the compounds are useful for the treatment of diseases and disorders related to the histamine H3 receptor.
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| 申请公布号 |
CA2473468(A1) |
申请公布日期 |
2003.08.07 |
| 申请号 |
CA20032473468 |
申请日期 |
2003.01.27 |
| 申请人 |
NOVO-NORDISK A/S |
发明人 |
PETTERSSON, INGRID;PESCHKE, BERND |
| 分类号 |
A61K31/4025;A61K31/4196;A61K31/454;A61P1/04;A61P1/08;A61P1/12;A61P1/16;A61P3/00;A61P3/04;A61P3/06;A61P3/10;A61P9/10;A61P9/12;A61P11/02;A61P11/06;A61P19/02;A61P25/00;A61P25/06;A61P25/08;A61P25/20;A61P25/24;A61P25/26;A61P25/28;A61P35/00;A61P37/00;A61P37/08;A61P43/00;C07D207/09;C07D211/26;C07D403/10;C07D405/06;C07D409/06;C07D521/00;(IPC1-7):C07D403/06;C07D401/06;C07D405/14;C07D409/14;A61K31/40;A61K31/402;A61K31/445;A61K31/452 |
主分类号 |
A61K31/4025 |
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