发明名称 N-ALKYLSULFONYL-SUBSTITUTED AMIDE DERIVATIVES
摘要 It is intended to provide ACC activity inhibitor which are efficacious in treating obesity, hyperlipemia and fat liver seemingly induced by obesity, glucose tolerance failure, diabetes and diabetic complications (diabetic peripheral neuropathy, diabetic nephropathy, diabetic retinopathy, diabetic great vessel disease, etc.) seemingly based on insulin resistance, hypertension and arteriosclerosis. N-Alkylsulfonyl-substituted amide derivatives, analogs thereof or pharmaceutically acceptable salts thereof have an efficacious ACC activity inhibitory effect.
申请公布号 WO03059871(A1) 申请公布日期 2003.07.24
申请号 WO2003JP00098 申请日期 2003.01.09
申请人 AJINOMOTO CO.,INC.;SUZUKI, NOBUYASU;NIHEI, YUKIO;ICHINOSE, HIDEHIRO;HATANAKA, TOSHIHIRO;MAEZONO, KATSUMI;OHSUMI, KOJI;KONDO, NOBUO 发明人 SUZUKI, NOBUYASU;NIHEI, YUKIO;ICHINOSE, HIDEHIRO;HATANAKA, TOSHIHIRO;MAEZONO, KATSUMI;OHSUMI, KOJI;KONDO, NOBUO
分类号 A61K45/00;A61K31/18;A61K31/426;A61K31/64;A61K38/28;A61P1/16;A61P3/04;A61P3/06;A61P3/10;A61P9/10;A61P9/12;A61P13/12;A61P25/00;A61P27/02;A61P43/00;C07C311/51;C07D277/30;(IPC1-7):C07C311/51;A61K31/427;A61K31/424;A61K31/381;A61K31/441;A61K31/443;A61K31/155;C07D213/82;C07D333/40;C07D417/04;C07D417/12;C07D271/06 主分类号 A61K45/00
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