发明名称 METHOD OF STABILIZATION FOR AMRUBICIN HYDROCHLORIDE
摘要 PROBLEM TO BE SOLVED: To provide a method which stabilizes (7S, 9S)-9-acetyl-9-amino-7-[(2- deoxy-β-D-erythro-pentapyranosil)oxy]-7,8,9,10-tetrahydro-6,11-dihydroxy-5,12- naphthacenediol hydrochloride (herein after abbreviated as amrubicin hydrochloride) expressed by general formula (1), more stably. SOLUTION: The method of stabilization for the amrubicin hydrochloride characteristically sets the water content of the amrubicin hydrochloride at 3-8 wt.%. COPYRIGHT: (C)2003,JPO
申请公布号 JP2003201297(A) 申请公布日期 2003.07.18
申请号 JP20020308101 申请日期 2002.10.23
申请人 SUMITOMO CHEM CO LTD;SUMITOMO PHARMACEUT CO LTD 发明人 TAKAHASHI KAZUHIKO;FUJIMOTO KOJI;YAMAUCHI YASUKO;OKABASHI YOSHITOKU
分类号 C07H15/252;A61K31/704;A61P35/00;(IPC1-7):C07H15/252 主分类号 C07H15/252
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