发明名称 DEAZAPURINES AND USES THEREOF
摘要 The present invention provides compounds having formula (I), wherein R<sb>1</sb>, R<sb>2</sb>, R<sb>3</sb> and n are as described generally and in classes and subclasses herein, and additionally provides pharmaceutical compositions thereof, and methods for the use thereof in the treatment of inflammatory or autoimmune and proliferative disorders and as inhibitors of cell adhesion molecule expression and inflammatory cytokine signal transduction generally.
申请公布号 WO03057696(A1) 申请公布日期 2003.07.17
申请号 WO2003US00366 申请日期 2003.01.07
申请人 EISAI CO. LTD.;DAUN, JANE;DAVIS, HEATHER, A.;GUSOVSKY, FABIAN;HISHINUMA, IEHARU;JIANG, YIMIN;KANEKO, TOSHIHIKO;KIKUCHI, KOUICHI;KOBAYASHI, SEIICHI;LESCARBEAU, ANDRE;LI, XIANG-LI;MURAMOTO, KENZO;OHI, NORIHITO;PESANT, MARC;SELETSKY, BORIS, M.;SOEJIMA, MOTOHIKO;YAO, YE;YOKOHAMA, HIROMITSU;ZHAO, JANET, Y.;ZHENG, WANJUN;TREMBLAY, LYNDA 发明人 DAUN, JANE;DAVIS, HEATHER, A.;GUSOVSKY, FABIAN;HISHINUMA, IEHARU;JIANG, YIMIN;KANEKO, TOSHIHIKO;KIKUCHI, KOUICHI;KOBAYASHI, SEIICHI;LESCARBEAU, ANDRE;LI, XIANG-LI;MURAMOTO, KENZO;OHI, NORIHITO;PESANT, MARC;SELETSKY, BORIS, M.;SOEJIMA, MOTOHIKO;YAO, YE;YOKOHAMA, HIROMITSU;ZHAO, JANET, Y.;ZHENG, WANJUN;TREMBLAY, LYNDA
分类号 A61K31/437;A61K31/444;A61K31/4545;A61K31/4709;A61K31/4725;A61K31/496;A61K31/5377;A61K31/541;A61K31/55;A61P1/04;A61P3/10;A61P7/04;A61P9/00;A61P11/02;A61P11/06;A61P13/12;A61P17/00;A61P17/04;A61P17/06;A61P19/02;A61P21/04;A61P25/00;A61P29/00;A61P31/12;A61P35/00;A61P37/00;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D471/04;C07D519/00;(IPC1-7):C07D471/04 主分类号 A61K31/437
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