发明名称 |
POLYMORPHS OF CLOPIDOGREL HYDROGENSULFATE |
摘要 |
Provided are new crystalline Forms III, IV, V and VI of clopidogrel hydrogensulfate and the amorphous form of clopidogrel hydrogensulfate, as well as their pharmaceutical compositions, and method of treatments with such compositions. Also provided are novel processes for preparation of clopidogrel hydrogensulfate Form I, Form II, Form III, Form IV, Form V, Form VI and amorphous form. |
申请公布号 |
WO03051362(A2) |
申请公布日期 |
2003.06.26 |
申请号 |
WO2002US40679 |
申请日期 |
2002.12.18 |
申请人 |
TEVA PHARMACEUTICAL INDUSTRIES LTD.;TEVA PHARMACEUTICALS USA, INC.;LIFSHITZ-LIRON, REVITAL;KOVALEVSKI-ISHAI, ETI;WIZEL, SHLOMIT;AVHAR-MAYDAN, SHARON;LIDOR-HADAS, RAMI |
发明人 |
LIFSHITZ-LIRON, REVITAL;KOVALEVSKI-ISHAI, ETI;WIZEL, SHLOMIT;AVHAR-MAYDAN, SHARON;LIDOR-HADAS, RAMI |
分类号 |
A61K31/4365;A61K31/44;A61P7/02;A61P9/10;C07D495/04;C07D515/02 |
主分类号 |
A61K31/4365 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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