发明名称 COMPOUNDS DERIVED FROM AN AMINE NUCLEUS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME
摘要 Compounds having the formula (I), are effective as inhibitors of IMPDH enzyme and/or serine protease Factor VIIa, wherein B is a monocyclic or bicyclic carbocyclic or heterocyclic ring, D is a monocyclic or bicyclic carbocyclic or heterocyclic ring except when A is a heterocyclic ring, then D is a heterocyclic ring system, R is hydrogen or C1-4alkyl, and A, R1, R2 and R4 are as defined in the specification.
申请公布号 WO03047512(A2) 申请公布日期 2003.06.12
申请号 WO2002US38038 申请日期 2002.11.27
申请人 BRISTOL-MYERS SQUIBB COMPANY;LIU, CHUNJIAN;DHAR, MURALI, T., G.;GU, HENRY, H.;IWANOWICZ, EDWIN, J.;LEFTHERIS, KATERINA;PITTS, WILLIAM, J.;HERPIN, TIMOTHY, F.;PI, ZULAN;BISACCHI, GREGORY, S. 发明人 LIU, CHUNJIAN;DHAR, MURALI, T., G.;GU, HENRY, H.;IWANOWICZ, EDWIN, J.;LEFTHERIS, KATERINA;PITTS, WILLIAM, J.;HERPIN, TIMOTHY, F.;PI, ZULAN;BISACCHI, GREGORY, S.
分类号 A61K45/06;C07D263/32;C07D263/48;C07D413/12;C07D413/14;C07D417/12;C07D521/00 主分类号 A61K45/06
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