摘要 |
PROBLEM TO BE SOLVED: To provide a method for producing an optically activeβ-arylamide compound usable for an intermediate for medicines or, agrochemicals in a high yield. SOLUTION: The optically activeβ-aryl amide compound can be produced for a short time and in a high yield by addition of a base such as potassium hydroxide, potassium carbonate, potassium hydrogen carbonate, potassium phosphate or the like when an arylboronic acid compound, its anhydride or arylboronic acid ester is reacted with anα,β-unsaturated amide in water or a water-containing solvent in the presence of a rhodium compound and an optically active phosphine compound. COPYRIGHT: (C)2003,JPO
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