发明名称 Method of preparing alkylated salicylamides via a dicarboxylate intermediate
摘要 The present invention relates to a method of preparing an alkylated salicylamide from a protected and activated salicylamide via a dicarboxylated salicylamide intermediate. The present invention also relates to dicarboxylic salicylamide delivery agent compounds for the delivery of active agents. Methods of administration are provided as well.
申请公布号 US2003096992(A1) 申请公布日期 2003.05.22
申请号 US20020239477 申请日期 2002.09.20
申请人 BERNADINO JOSEPH N.;O'TOOLE DORIS C.;BAY WILLIAM E. 发明人 BERNADINO JOSEPH N.;O'TOOLE DORIS C.;BAY WILLIAM E.
分类号 C07D265/36;A61K45/00;A61K47/16;A61P1/04;A61P3/00;A61P3/02;A61P5/06;A61P7/00;A61P7/02;A61P9/00;A61P9/08;A61P9/12;A61P11/06;A61P13/00;A61P15/00;A61P19/08;A61P19/10;A61P31/00;A61P35/00;A61P37/02;A61P37/08;A61P43/00;C07C231/12;C07C235/60;C07C269/00;C07C271/64;C07D265/22;C07D265/26;(IPC1-7):C07D265/12;C07C255/44;C07C235/84 主分类号 C07D265/36
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