| 发明名称 |
Selective androgen receptor modulator, method of its identification, its construction, and use |
| 摘要 |
<p>Selective androgen receptor modulators (SARMs) having antagonist activity in hormone-dependent tumors while exhibiting no activity or agonist activity against other nontumor tissues containing the androgen receptor as well as methods for identifying, designing and using SARMs are provided.</p> |
| 申请公布号 |
CZ20024214(A3) |
申请公布日期 |
2003.04.16 |
| 申请号 |
CZ20020004214 |
申请日期 |
2001.06.20 |
| 申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
SALVATI MARK E.;GOTTARDIS MARCO M.;KRYSTEK STANLEY R. JR.;ATTAR RICARDO M.;SACK JOHN S. |
| 分类号 |
G01N33/483;A61K31/00;A61K31/407;A61K31/4155;A61K31/416;A61K31/4196;A61K31/42;A61K31/433;A61K31/4439;A61K31/4709;A61K31/4995;A61K31/506;A61K31/655;A61K31/675;A61K45/00;A61P5/28;A61P13/08;A61P35/00;C07D471/18;C07D487/08;C07D487/18;C07D491/08;C07D491/18;C07D491/22;C07D493/18;C07D495/18;C07D519/00;C07K14/72;C12Q1/02;G01N33/15;G01N33/50;G01N33/53;(IPC1-7):A61K31/407;C07D201/00 |
主分类号 |
G01N33/483 |
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