发明名称 |
3-`HYDROXY-(-4-TRIFLUOROMETHYLPHENYL)-METHYL-7-SPIROCYCLOBUTYL-5,6,7,8-TETRAHYDROQUINOLIN-5-OL DERIVATIVES AND THE USE OF THE SAME AS CHOLESTEROL ESTER TRANSFER PROTEIN (CETP) INHIBITORS |
摘要 |
The invention relates to substituted tetrahydroquinoline derivatives of formula (I), wherein A represents a radical (a), (b), (c), (d), (e), (f), (g ), (h) or -(CH2)2CH3 and B represents a radical (f) or (h), and to the salts of the same. The invention also relates to a method for producing said substanc es and to the use thereof in pharmaceuticals.
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申请公布号 |
CA2462030(A1) |
申请公布日期 |
2003.04.10 |
申请号 |
CA20022462030 |
申请日期 |
2002.09.18 |
申请人 |
BAYER HEALTHCARE AG |
发明人 |
KELDENICH, JOERG;PAULSEN, HOLGER;GIELEN, HEIKE;SCHMECK, CARSTEN;SCHMIDT, DELF;SIEGEL, STEPHAN;BISCHOFF, HILMAR;RAABE, MARTIN;FAESTE, CHRISTIANE;GOLDMANN, SIEGFRIED |
分类号 |
C07D215/20;A61K31/47;A61K31/4709;A61P3/04;A61P3/06;A61P9/00;A61P9/10;A61P25/28;A61P43/00;C07D221/20;C07D409/04;(IPC1-7):C07D409/04;A61K31/470;A61K31/474 |
主分类号 |
C07D215/20 |
代理机构 |
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