发明名称 |
11BETA-HALOGEN-7ALPHA-SUBSTITUTED ESTRATRIENES, METOD FOR PRODUCING PHARMACEUTICAL PREPARATIONS CONTAINING SAID 11BETA-HALOGEN-7ALPHA- SUBSTITUTED ESTRATRIENES AND USE OF THE SAME FOR PRODUCING MEDICAMENTS |
摘要 |
This invention describes the new 11beta-halogen-7alpha-substituted estratrienes of general formula I in which R<11 >is a fluorine or chlorine atom, and the other substituents have the meanings that are explained in more detail in the description. The compounds have antiestrogenic properties or tissue-selective estrogenic properties and are suitable for the production of pharmaceutical agents.
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申请公布号 |
US2003069434(A1) |
申请公布日期 |
2003.04.10 |
申请号 |
US19990380413 |
申请日期 |
1999.12.02 |
申请人 |
BOHLMANN ROLF;HEINRICH NIKOLAUS;HOFMEISTER HELMUT;KROLL JORG;KUNZER HERMANN;SAUER GERHARD;ZORN LUDWIG;FRITZEMEIER KARL-HEINRICH;LESSL MONIKA;LICHTNER ROSEMARIE;NISHINO YUKISHIGE;PARCZYK KARSTEN;SCHNEIDER MARTIN |
发明人 |
BOHLMANN ROLF;HEINRICH NIKOLAUS;HOFMEISTER HELMUT;KROLL JORG;KUNZER HERMANN;SAUER GERHARD;ZORN LUDWIG;FRITZEMEIER KARL-HEINRICH;LESSL MONIKA;LICHTNER ROSEMARIE;NISHINO YUKISHIGE;PARCZYK KARSTEN;SCHNEIDER MARTIN |
分类号 |
A61K31/565;A61K31/58;A61P5/32;A61P43/00;C07J31/00;C07J41/00;C07J43/00;(IPC1-7):C07J1/00;A61K31/56 |
主分类号 |
A61K31/565 |
代理机构 |
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