发明名称 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors
摘要 Prodrugs of COX-2 inhibitors and methods of their preparation are described. The prodrugs of COX-2 inhibitors are described as being useful in treating inflammation and inflammation-related disorders.
申请公布号 US2003069287(A1) 申请公布日期 2003.04.10
申请号 US20020178697 申请日期 2002.06.24
申请人 PHARMACIA CORPORATION 发明人 TALLEY JOHN J.;MALECHA JAMES W.;BERTENSHAW STEPHEN;GRANETO MATTHEW J.;CARTER JEFFERY S.;LI JINGLIN;NAGARAJAN SRINIVASAN;BROWN DAVID L.;ROGIER DONALD J.;PENNING THOMAS D.;KHANNA ISH K.;XU XIANGDONG;WEIER RICHARD M.
分类号 C07D233/64;A61K31/00;A61K31/18;A61K31/34;A61K31/341;A61K31/365;A61K31/40;A61K31/415;A61K31/4162;A61K31/4164;A61K31/42;A61K31/421;A61K31/44;A61K31/4427;A61K31/4439;A61K31/635;A61P1/02;A61P1/04;A61P3/10;A61P5/16;A61P7/06;A61P9/10;A61P11/02;A61P11/06;A61P11/08;A61P13/12;A61P15/06;A61P17/02;A61P17/04;A61P17/06;A61P19/02;A61P19/08;A61P21/00;A61P21/04;A61P25/00;A61P25/04;A61P25/28;A61P27/02;A61P27/12;A61P29/00;A61P29/02;A61P31/12;A61P35/00;A61P37/00;A61P43/00;C07C311/16;C07C311/39;C07C311/51;C07D;C07D207/32;C07D207/327;C07D207/33;C07D231/12;C07D233/54;C07D233/62;C07D261/08;C07D263/32;C07D307/46;C07D307/58;C07D401/04;C07D417/04;C07D495/04;(IPC1-7):A61K31/44;A61K31/402 主分类号 C07D233/64
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