发明名称 6-MEMBERED UNSATURATED HETEROCYCLIC COMPOUNDS USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE
摘要 The present invention relates to compounds, and prodrugs thereof, compositio n and methods useful for preventing and treating thrombotic conditions in mammals. The compounds of the present invention, and prodrugs thereof, selectively inhibit certain proteases of the coagulation cascade.
申请公布号 CA2462647(A1) 申请公布日期 2003.04.10
申请号 CA20022462647 申请日期 2002.10.03
申请人 PHARMACIA CORPORATION 发明人 WOOD, RHONDA S.;ABBAS, ZAHEER;ZENG, QINGPING;RUEPPEL, MELVIN L.;HAYES, MICHAEL J.;SULEYMANOV, OSMAN D.;SNYDER, JEFFREY S.;SZALONY, JIM;JONES, DARIN E.;SALYERS, ANITA;TOTH, MIHALY V.;MOORMANN, ALAN E.;CASE, BRENDA;NEUMANN, WILLIAM L.;HUANG, HORNG-CHIH;LONG, SCOTT;WEBBER, RONALD K.;TRUJILLO, JOHN;WEI, HUANG;KUSTURIN, CARRIE L.;HAYAT, RAHMAN K.;SCHOLTEN, JEFFREY A.;SOUTH, MICHAEL S.;GARLAND, DANNY J.;SAMPLE, KIRBY R.;NICHOLSON, NANCY S.;PARLOW, JOHN J.;FENTON, RICKY L.;SCHWEITZER, BARBARA A.
分类号 C07D239/47;A61K31/4965;A61K31/497;A61K31/513;A61K31/5377;A61K31/616;A61K45/00;A61P7/02;A61P43/00;C07C257/18;C07D207/32;C07D211/56;C07D211/98;C07D213/74;C07D231/38;C07D231/48;C07D237/04;C07D239/10;C07D239/22;C07D241/04;C07D241/20;C07D249/14;C07D253/06;C07D253/075;C07D263/48;C07D265/02;C07D277/42;C07D307/22;C07D333/36;C07D401/12;C07D403/04;C07D403/10;C07D409/12;C07D413/12;C07D471/04;(IPC1-7):C07D239/47;C07D403/12;A61K31/496 主分类号 C07D239/47
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