发明名称 Tetracyclic azepinoindole compounds as 5-HT receptor ligands.
摘要 The present invention provides compounds of formula (I), wherein R2 is hydrogen, C1-7alkyl, C1-7alkanoyl, arylcarbonyl, aryl, (aryl)C1-7alkyl, C1-7alkoxycarbonyl, aryloxycarbonyl, arylsulfonyl, or (aryl)C1-7alkoxycarbonyl; X and Y together are 2, 3 or 4 membered saturated or partially unsaturated chain. These compounds are 5-HT ligands, and are useful for treating diseases wherein modulation of 5-HT activity is desired.
申请公布号 ZA200108636(B) 申请公布日期 2003.02.19
申请号 ZA20010008636 申请日期 2001.10.19
申请人 PHARMACIA & UPJOHN COMPANY 发明人 JACKSON B. HESTER;E. JON JACOBSEN;BRAD A. ACKER;KRISTINE E. FRANK;BRUCE N. ROGERS;MICHAEL DALTON ENNIS;SUSAN L. VAN DER VELDE
分类号 C07D487/04;A61K31/395;A61K31/55;A61P1/00;A61P1/08;A61P3/04;A61P9/00;A61P9/12;A61P13/00;A61P15/00;A61P15/10;A61P21/00;A61P25/00;A61P25/02;A61P25/04;A61P25/06;A61P25/14;A61P25/18;A61P25/22;A61P25/30;A61P37/02;A61P43/00;C07D471/14;C07D471/16;C07D498/16;C07D513/16 主分类号 C07D487/04
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