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发明名称
BENZIMIDAZO[4,5-f]ISOQUINOLINONE DERIVATIVES
摘要
Benzimidazo[4,5-f]isoquinolinone derivatives are inhibitors of Janus protein tyrosine kinases (Jak), and as such are useful as immunosuppressants, and in the treatment of diseases including asthma, allergies, autoimmune diseases .
申请公布号
WO03011285(A1)
申请公布日期
2003.02.13
申请号
WO2002US23876
申请日期
2002.07.26
申请人
MERCK & CO., INC.;GOULET, JOUNG, L.;HONG, XINGFANG;SINCLAIR, PETER, J.;THOMPSON, JAMES, E.;CUBBON, ROSE, M.;CUMMINGS, RICHARD, T.
发明人
GOULET, JOUNG, L.;HONG, XINGFANG;SINCLAIR, PETER, J.;THOMPSON, JAMES, E.;CUBBON, ROSE, M.;CUMMINGS, RICHARD, T.
分类号
A61K31/4745;A61P3/10;A61P5/14;A61P7/10;A61P11/02;A61P11/06;A61P17/04;A61P21/04;A61P29/00;A61P35/00;A61P35/02;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D471/04;C07D471/14;(IPC1-7):A61K31/407;C07D215/18;C07D215/20;C07D215/22
主分类号
A61K31/4745
代理机构
代理人
主权项
地址
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