发明名称 NOVEL 2 H -PYRIDAZINE-3-ONE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND A PROCESS FOR THE PREPARATION OF THE ACTIVE INGREDIENT
摘要 The invention refers to novel 2H-pyridazine-3-one derivatives of the formula I, pharmaceutical compositions containing the same and a process for the preparation of the active ingredient. The novel compounds possess neuroleptic effect and can be used, primarily, for the treatment of schizophrenia. In formula I, R stands for a hydrogen atom or a C1-4 alkyl group, X and Y represent, independently, a hydrogen atom, a halogen atom or a group of the formula II, with the proviso that one of X and Y means always a group of the formula II, and then the other one stands for a hydrogen atom or a halogen atom, wherein in formula II n has a value of 1 or 2.
申请公布号 WO03010166(A1) 申请公布日期 2003.02.06
申请号 WO2002HU00072 申请日期 2002.07.24
申请人 EGIS GYOGYSZERGYAR RT.;BARKOCZY, JOZSEF;KOTAY NAGY, PETER;SIMIG, GYULA;LEVAY, GYOERGY;GACSALYI, ISTVAN;EGYED, ANDRAS;RACZNE BAJNOGEL, JUDIT;PALLAGI, KATALIN;SCHMIDT, EVA;SZENASI, GABOR;MIKLOSNE KOVACS, ANIKO;WELLMANN, JANOS 发明人 BARKOCZY, JOZSEF;KOTAY NAGY, PETER;SIMIG, GYULA;LEVAY, GYOERGY;GACSALYI, ISTVAN;EGYED, ANDRAS;RACZNE BAJNOGEL, JUDIT;PALLAGI, KATALIN;SCHMIDT, EVA;SZENASI, GABOR;MIKLOSNE KOVACS, ANIKO;WELLMANN, JANOS
分类号 A61K31/501;A61P25/18;A61P25/22;A61P25/24;C07D413/14;(IPC1-7):C07D413/14;A61K31/50 主分类号 A61K31/501
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