发明名称 NOVEL BRANCHED SUBSTITUTED AMINO DERIVATIVES OF 3AMINO1PHENYLH.
摘要 <p>The invention relates to compounds of general formula (I), wherein in particular, R1, R2, and R3 represent, each independently of each other, hydrogen, a halogen atom; a (C1C5)alkyl; a (C1C5)alkoxy; a trifluoromethyl or a group SR, wherein R represents a (C1C5)alkyl; R4, R5 represents a (C1C5)alkyl; an alkynyl with 3 to 5 carbon atoms; a (C3C5)cycloalkyl or an RaX(C1C2)alkyl group wherein Ra represents a (C1C3)alkyl and X represents O; R6 represents CHR7R8 wherein R7 represents a phenyl group which can be substituted by one or more radicals Z in position 3, 4 and 5, with Z representing a halogen; a (C1C5)alkyl; a (C1C5)alkylX or (C1C3)alkylX(C1C2)alkyl or X represents O; or a methylenedioxy group; and R8 represents a (C1C6)alkyl; a (C3C5)cycloalkyl(C1C3)alkyl; (C1C3)alkylX(C1C3)alkyle wherein X represents O. These compounds are suitable for CRF receptors.</p>
申请公布号 MXPA02006033(A) 申请公布日期 2003.01.28
申请号 MX2002PA06033 申请日期 2000.12.14
申请人 SANOFI-SYNTHELABO 发明人 GESLIN, MICHEL
分类号 A61K31/4196;A61P1/14;A61P15/10;A61P25/00;A61P25/08;A61P25/22;A61P25/24;A61P25/28;A61P29/00;A61P35/00;A61P43/00;B29C44/12;C07D249/14;C07D405/12;(IPC1-7):C07D249/14 主分类号 A61K31/4196
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