发明名称 ALIPHATIC NITROGEN-CONTAINING FIVE-MEMBERED RING COMPOUND
摘要 PROBLEM TO BE SOLVED: To provide a new aliphatic nitrogen-containing five-membered ring compound having excellent DPPIV inhibitory action. SOLUTION: This compound is an aliphatic nitrogen-containing five-membered ring compound represented by the formula [I] [wherein, A is CH2 or S; R<1> is H, a lower alkyl, a hydroxy lower alkyl or a lower alkoxy lower alkyl; X is N(R<3> ), O or CO; R<3> is H or a lower alkyl; and R<2> is (1) a (substituted)cyclic group or (2) a (substituted)amino group.] or a pharmacologically permissible salt of the compound, and the method for producing the compound is also provided.
申请公布号 JP2002356471(A) 申请公布日期 2002.12.13
申请号 JP20010309558 申请日期 2001.10.05
申请人 TANABE SEIYAKU CO LTD 发明人 YASUDA KOUSUKE;MORIMOTO HIROSHI;KAWANAMI SABURO;HIKODA MASAKATSU;MATSUMOTO TAKESHI;ARAKAWA KENJI
分类号 C07D277/12;A61K31/40;A61K31/4035;A61K31/41;A61K31/423;A61K31/426;A61K31/427;A61K31/428;A61K31/433;A61K31/4439;A61K31/454;A61K31/4725;A61K31/496;A61K31/497;A61K31/498;A61K31/501;A61K31/506;A61K31/519;A61K31/5377;A61K31/541;A61K31/55;A61P3/10;A61P19/02;A61P19/10;A61P29/00;A61P37/02;A61P43/00;C07D207/16;C07D277/20;C07D277/44;C07D401/12;C07D401/14;C07D403/12;C07D405/12;C07D405/14;C07D409/12;C07D409/14;C07D413/12;C07D417/12;C07D471/04;C07D491/048;C07D495/04;(IPC1-7):C07D207/16;A61K31/403;A61K31/443;A61K31/472;A61K31/537 主分类号 C07D277/12
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